A selective estrogen receptor modulator 50 mg


≥98% pure A selective estrogen receptor modulator 50 mg



Raloxifene is a selective estrogen receptor modulator (SERM) that binds to the estrogen receptor with an IC50 value of 0.4 nM.1 It exhibits estrogenic activity in bone cells without stimulating breast or uterine tissues.2 Raloxifene guards endothelial cells obtained from rat aortic rings against oxidative insult (1 µM) and lowers serum cholesterol in ovariectomized rodents (ED50 = 0.2 mg/kg).2,3 Raloxifene also inhibits the voltage-gated potassium channel Kv4.3 in an estrogen-independent manner (IC50 = 2 µM).4 Formulations containing raloxifene have been shown to reduce bone resorption and promote bone formation in post-menopausal women.5
WARNING This product is not for human or veterinary use.


There are no reviews yet.

Be the first to review “A selective estrogen receptor modulator 50 mg”

Your email address will not be published. Required fields are marked *

Got something to discuss?